Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-1' and Ligand = 'BDBM50449237'
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Yerevan State University

Curated by ChEMBL
LigandPNGBDBM50449237(CHEMBL3128141)
Affinity DataIC50:  600nMAssay Description:Inhibition of 20s immunoproteasome beta 1 subunit caspase-like activity in human blood monocytes using Z-LLE-betaNA as substrate at 2 uM preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Yerevan State University

Curated by ChEMBL
LigandPNGBDBM50449237(CHEMBL3128141)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of 20s proteasome beta 1 subunit caspase-like activity in human HeLa cells using Z-nLPnLD as substrate after 17 hrs by chemiluminescence a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed