Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50059876'
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against rat brain farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  20nMAssay Description:Inhibition of rat brain farnesyltransferase in 30 mM potassium phosphate bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  76nMAssay Description:In vitro inhibition of rat farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  76nMAssay Description:Inhibition of rat brain farnesyltransferase in 5 mM potassium phosphate and 50 mM HEPES bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  420nMAssay Description:Inhibition of Ras-processing in H-Ras transformed NIH3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat brain farnesyltransferase in 50 mM HEPES bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed