Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50106865'
LigandPNGBDBM50106865(1-(3-Benzo[1,3]dioxol-5-ylmethyl-3H-imidazol-4-ylm...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of farnesyltransferase activity against H-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106865(1-(3-Benzo[1,3]dioxol-5-ylmethyl-3H-imidazol-4-ylm...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of farnesyltransferase activity against K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed