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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase B-raf' and Ligand = 'BDBM50344475'
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50344475(2-(4-(2,4-dihydroindeno[1,2-c]pyrazol-6-yl)-3-(pyr...)
Affinity DataIC50:  72.5nMAssay Description:Inhibition of B-RafMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50344475(2-(4-(2,4-dihydroindeno[1,2-c]pyrazol-6-yl)-3-(pyr...)
Affinity DataIC50:  8.16E+3nMAssay Description:Inhibition of B-Raf-mediated ERK phosphorylation in cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed