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Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk2' and Ligand = 'BDBM50363645'
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50363645(DEBROMOHYMENIALDISINE)
Affinity DataIC50:  180nMAssay Description:Antagonist activity in phenoxybenzamine-treated rat by Pressor assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50363645(DEBROMOHYMENIALDISINE)
Affinity DataIC50:  183nMAssay Description:Antagonist activity in rat uterus by uterotonic assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50363645(DEBROMOHYMENIALDISINE)
Affinity DataIC50:  183nMAssay Description:Inhibition of human Chk2 using STK1 as substrate after 10 mins by HTRF assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50363645(DEBROMOHYMENIALDISINE)
Affinity DataIC50:  183nMAssay Description:Inhibition of CHK2 (unknown origin) using polypeptide substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50363645(DEBROMOHYMENIALDISINE)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Chk2Checked by AuthorMore data for this Ligand-Target Pair