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Found 1 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1B1' and Ligand = 'BDBM50581546'
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50581546(CHEMBL5084416)
Affinity DataEC50: >2.20E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed