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Found 7 Enz. Inhib. hit(s) with Target = 'Sortase family protein' and Ligand = 'BDBM50590366'
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataKi:  2.45E+3nMAssay Description:Irreversible inhibition of recombinant Staphylococcus aureus sortase A deltaN24 expressed in Escherichia coli BL21(DE3) cells using Abz-LPATG-Dnp as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  300nMAssay Description:Irreversible inhibition of recombinant Staphylococcus aureus sortase A deltaN24 expressed in Escherichia coli BL21(DE3) cells using Abz-LPATG-Dnp as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant Staphylococcus aureus sortase A deltaN24 transpeptidation expressed in Escherichia coli BL21 (DE3) cells using Abz-LPATG-Dn...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  400nMAssay Description:Irreversible inhibition of recombinant Staphylococcus aureus sortase A deltaN24 expressed in Escherichia coli BL21(DE3) cells using Abz-LPATG-Dnp as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  500nMAssay Description:Irreversible inhibition of recombinant Staphylococcus aureus sortase A deltaN24 expressed in Escherichia coli BL21(DE3) cells using Abz-LPATG-Dnp as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  1.10E+3nMAssay Description:Irreversible inhibition of recombinant Staphylococcus aureus sortase A deltaN24 expressed in Escherichia coli BL21(DE3) cells using Abz-LPATG-Dnp as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSortase family protein(Staphylococcus aureus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50590366(CHEMBL5174805)
Affinity DataIC50:  2.65E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus sortase A deltaN24 transpeptidation expressed in Escherichia coli BL21 (DE3) cells using IsdA64 to 32...More data for this Ligand-Target Pair
In DepthDetails PubMed