TargetSphingosine kinase 1(Homo sapiens (Human))
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.33E+3nMAssay Description:Competitive inhibition of recombinant sphingosine kinase 1 using D-erythro-sphingosine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Pennsylvania State University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant His6x-tagged human SphK1 expressed in HEK293 cells assessed as reduction in S1P formation using D-erythro-sphingosine as su...More data for this Ligand-Target Pair