Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Steroidogenic factor 1' and Ligand = 'BDBM50418303'
TargetSteroidogenic factor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of 6N-FAM from SF1 LBD (218 to 461 residues) (unknown origin) expressed in Escherichia coli BL21 pLysS by competitive binding based fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to human SF1 LBD (218 to 461 residues) expressed in Escherichia coli BL21 by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed