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Found 3 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM50366524'
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366524(ESTRONE | ESTROPIPATE | Estrone 3-sulfate | Estron...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibitory activity against steroid sulfatase (STS) desulfation of 4-MUSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366524(ESTRONE | ESTROPIPATE | Estrone 3-sulfate | Estron...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of steroid sulfatase activity of JEG-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50366524(ESTRONE | ESTROPIPATE | Estrone 3-sulfate | Estron...)
Affinity DataIC50:  7.60E+3nMAssay Description:Estrone sulfatase activity against homogenized human JEG-3 cells was determined by measuring the [3H]E1 obtained from [3H]E1SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed