Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50460759'
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Mannheim University Of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  5.89E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Mannheim University Of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  7.10E+3nMAssay Description:Activation of rat TRPV1 transfected in HEK293 cells assessed as increase in calcium influx in presence of capsaicin by FURA-2-AM dye based fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Mannheim University Of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  5.93E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed