Found 1 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50558639'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Mannheim University Of Applied Sciences
Curated by ChEMBL
Mannheim University Of Applied Sciences
Curated by ChEMBL
Affinity DataEC50: 4.59E+4nMAssay Description:Activation of rat TRPV1 transfected in HEK293 cells assessed as increase in calcium influx in presence of capsaicin by FURA-2-AM dye based fluorescen...More data for this Ligand-Target Pair