Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein phosphatase non-receptor type 1' and Ligand = 'BDBM14244'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM14244(4,5-dibromo-3-(carboxymethoxy)thiophene-2-carboxyl...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of PTP1B assessed as pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM14244(4,5-dibromo-3-(carboxymethoxy)thiophene-2-carboxyl...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of PTP1B assessed as pNPP hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed