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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosyl-DNA phosphodiesterase 1' and Ligand = 'BDBM60991'
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue Research Foundation

US Patent
LigandPNGBDBM60991(BDBM50425048 | US9402842, 14)
Affinity DataIC50:  6.10E+4nMpH: 7.5 T: 2°CAssay Description:A 5′-[32P]-labeled single-stranded DNA oligonucleotide containing a 3′-phosphotyrosine (N14Y) was generated as described by Dexheimer et ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue Research Foundation

US Patent
LigandPNGBDBM60991(BDBM50425048 | US9402842, 14)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of recombinant Tdp1 (unknown origin) using 5'-[32P]-labeled single-stranded DNA oligonucleotide containing 3'-phosphotyrosine as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue Research Foundation

US Patent
LigandPNGBDBM60991(BDBM50425048 | US9402842, 14)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to recombinant Tdp1 (unknown origin) using 3'-phosphate(GATCTAAAAGACTT) as substrate by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed