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TargetEukaryotic initiation factor 4A-I(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50610971(CHEMBL5290937)
Affinity DataEC50:  2.75E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataKd:  14nMAssay Description:Binding affinity to 6His-tagged BRD3-BD1 (unknown origin) by MST assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataKd:  149nMAssay Description:Binding affinity to 6His-tagged BRD3-BD2 (unknown origin) by MST assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1A (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1-like(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1L (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA2 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  334nMAssay Description:Binding affinity to HspA5 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 6(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA6 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA8 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  7.48E+3nMAssay Description:Binding affinity to HspA9 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to human partial length BRD4 BD2 (K333 to E460 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to human partial length BRDT BD2 (K250 to E382 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 7.10nMAssay Description:Binding affinity to human partial length BRD3 BD1 (P24 to E144 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 7.60nMAssay Description:Binding affinity to human partial length BRD3 BD2 (G306 to P416 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 9.30nMAssay Description:Binding affinity to human partial length BRD2 BD2 (E348to D455 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 18nMAssay Description:Binding affinity to human partial length BRD4 BD1 (N44 to E168 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50: 18nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50: 19nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616257(CHEMBL3605566)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616258(CHEMBL4074906)
Affinity DataIC50: 48nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 56nMAssay Description:Binding affinity to human partial length BRD4 BD1 (N44 to E168 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616263(CHEMBL4082632)
Affinity DataIC50: 60nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 69nMAssay Description:Binding affinity to human partial length BRD3 BD1 (P24 to E144 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616257(CHEMBL3605566)
Affinity DataIC50: 90nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 103nMAssay Description:Binding affinity to human partial length BRD2 BD1 (K71 to N194 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 108nMAssay Description:Binding affinity to human partial length BRD3 BD2 (G306 to P416 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 119nMAssay Description:Binding affinity to human partial length BRDT BD2 (K250 to E382 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 131nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 142nMAssay Description:Binding affinity to human partial length BRD4 BD2 (K333 to E460 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616258(CHEMBL4074906)
Affinity DataIC50: 210nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616263(CHEMBL4082632)
Affinity DataIC50: 235nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 244nMAssay Description:Binding affinity to human partial length BRD2 BD2 (E348to D455 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University

Curated by ChEMBL
LigandPNGBDBM42034(4-(3-nitro-4-oxidanyl-phenyl)-3a,4,5,9b-tetrahydro...)
Affinity DataIC50: 250nMAssay Description:Inhibition of Escherichia coli GroEL/GroES using Escherichia coli GroEL expressed in Escherichia coli DH5alpha cells and Escherichia coli GroES expre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 262nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616259(CHEMBL5412959)
Affinity DataIC50: 281nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 294nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 403nMAssay Description:Binding affinity to human partial length BRDT BD1 (N21 to E137 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University

Curated by ChEMBL
LigandPNGBDBM42034(4-(3-nitro-4-oxidanyl-phenyl)-3a,4,5,9b-tetrahydro...)
Affinity DataIC50: 470nMAssay Description:Inhibition of Escherichia coli GroEL/GroES using Escherichia coli GroEL expressed in Escherichia coli DH5alpha cells and Escherichia coli GroES expre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617266(CHEMBL5418499)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617268(CHEMBL5415571)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 6(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA6 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 510nMAssay Description:Binding affinity to human partial length BRDT BD1 (N21 to E137 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50437341(WITHANOLIDE E)
Affinity DataIC50: 556nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50495801(CHEMBL3115911)
Affinity DataIC50: 580nMAssay Description:Inhibition of Escherichia coli GroEL/GroES using Escherichia coli GroEL expressed in Escherichia coli DH5alpha cells and Escherichia coli GroES expre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617261(CHEMBL5414287)
Affinity DataIC50: 590nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50495801(CHEMBL3115911)
Affinity DataIC50: 690nMAssay Description:Inhibition of Escherichia coli GroEL/GroES using Escherichia coli GroEL expressed in Escherichia coli DH5alpha cells and Escherichia coli GroES expre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 700nMAssay Description:Inhibition of HspA2 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617277(CHEMBL5419391)
Affinity DataIC50: 700nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50437341(WITHANOLIDE E)
Affinity DataIC50: 720nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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