Report error Found 1833 with Last Name = 'corelli' and Initial = 'f'
Affinity DataEC50: 1.14E+3nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 318nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 371nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 1.53E+3nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 197nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 252nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 3.15E+3nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 2.67E+4nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 1.45E+3nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 880nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 2.08E+3nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 1.18E+3nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 590nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 391nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 628nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 6.20nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membrane assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liq...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membrane assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liq...More data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membrane assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liq...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membrane assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liq...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataEC50: 398nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liqu...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liqu...More data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liqu...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liqu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Activation of human TRPV1 expressed in HEK293 cells assessed as calcium influx preincubated for 5 mins by Fluo-4AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 1.11E+4nMAssay Description:Activation of rat recombinant TRPA1 expressed in HEK293 cells assessed as calcium influx preincubated for 5 mins by Fluo-4AM dye based fluorescence a...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Magna Gracia University
Curated by ChEMBL
Magna Gracia University
Curated by ChEMBL
Affinity DataEC50: 3.5nMAssay Description:Agonist activity at rat recombinant TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 1.88E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 234nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 1.15E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 676nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 741nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 841nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 61nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 108nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 109nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 870nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
