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Found 20 with Last Name = 'pérez-fernández' and Initial = 'r'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataKi:  400nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataKi:  5.25E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135847(Bicyclic Guanidinium Subunit | CHEMBL404936)
Affinity DataKi:  7.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50:  1.24nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397221(CHEMBL2172537)
Affinity DataIC50:  15.7nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397223(CHEMBL2172539)
Affinity DataIC50:  20.9nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397222(CHEMBL2172538)
Affinity DataIC50:  27.3nMAssay Description:Binding affinity to VDR assessed as inhibition of fluorescent ligand by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135843(Bicyclic Guanidinium Subunit | CHEMBL216653)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135843(Bicyclic Guanidinium Subunit | CHEMBL216653)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135846(Bicyclic Guanidinium Subunit | CHEMBL428283)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135847(Bicyclic Guanidinium Subunit | CHEMBL404936)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£noma de Madrid

Curated by ChEMBL
LigandPNGBDBM50135848(Bicyclic Guanidinium Subunit | CHEMBL414980)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  3.28nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397223(CHEMBL2172539)
Affinity DataEC50:  8.19nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397222(CHEMBL2172538)
Affinity DataEC50:  9.04nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50397221(CHEMBL2172537)
Affinity DataEC50:  5.74nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed