TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 0.0960nMAssay Description:Binding affinity to CLK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 0.0960nMAssay Description:Binding affinity to CLK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 0.510nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 0.900nMAssay Description:Inhibition of human partial length CLK2 (D144/R498) expressed in bacterial system by DiscoveryX Kinomescan binding assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 8.20nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 8.20nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 8.20nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to human CLK2More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Average Binding Constant for CLK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding affinity to CLK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to recombinant human CLK2 (D144 to R498 residues) expressed in bacterial expression system by KinomeScan assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to CLK2More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 43nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 44nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 44nMAssay Description:Binding affinity to CLK2More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 59nMAssay Description:Binding affinity to human Clk2 More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 80nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 82nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 93nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 95nMAssay Description:Binding affinity to Clk2 assessed as dissociation constantMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Average Binding Constant for CLK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 220nMAssay Description:Binding affinity to wild-type human partial length CLK2 (D144 to R498 residues) expressed in bacterial expression system measured after 1 hr by compe...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Average Binding Constant for CLK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 318nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged CLK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Binding affinity to human Clk2 More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 360nMAssay Description:Binding affinity to CLK2More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 380nMAssay Description:Binding affinity to human Clk2 More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 396nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged CLK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 410nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 420nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 420nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 420nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 430nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Inhibition of wild-type human partial length CLK2 (D144 to R498 residues) expressed in bacterial expression system by Kinomescan method relative to c...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding affinity to recombinant human CLK2 (D144 to R498 residues) expressed in bacterial expression system by KinomeScan assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Average Binding Constant for CLK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair