Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]DAMGO from calf thalamus membrane MOP by competitive binding assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DAMGO from calf thalamus membrane MOP by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.29nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity of the compound towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity of the compound towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 25.2nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 25.2nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 27.7nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 40.6nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity towards opioid receptor mu 2More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinity of the compound towards opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 91.6nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Activity of the compound was evaluated by inhibition of the binding of 0.8 nM [3H]- DAMGO at Opioid receptor mu 1 binding siteMore data for this Ligand-Target Pair
