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Found 30 of ki for UniProtKB: P16177
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290462(CHEMBL305119 | potassium 2N-[1-benzyl(methyl)carba...)
Affinity DataKi:  5nMAssay Description:Binding affinity of the compound for NK-3 receptor was determined in vitro using isolated rat portal vein.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290461(CHEMBL65468 | potassium 3,5-di(trifluoromethyl)ben...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity of the compound for NK-3 receptor was determined in vitro using isolated rat portal vein.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081194(CHEMBL3422009 | US10544150, Compound 156)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081194(CHEMBL3422009 | US10544150, Compound 156)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081198(CHEMBL3422018 | US10065961, Compound 24 | US947581...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081198(CHEMBL3422018 | US10065961, Compound 24 | US947581...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081198(CHEMBL3422018 | US10065961, Compound 24 | US947581...)
Affinity DataKi:  22nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081196(CHEMBL3422015 | US10065961, Compound 13 | US106832...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081196(CHEMBL3422015 | US10065961, Compound 13 | US106832...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)
Affinity DataKi:  57nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081195(CHEMBL3422010 | US10065961, Compound 1 | US1068329...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081195(CHEMBL3422010 | US10065961, Compound 1 | US1068329...)
Affinity DataKi:  76nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081195(CHEMBL3422010 | US10065961, Compound 1 | US1068329...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50112180(CHEMBL3608688 | US10030025, Compound 41 | US108367...)
Affinity DataKi:  85nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081197(CHEMBL3422017 | US10065961, Compound 23 | US106832...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50081197(CHEMBL3422017 | US10065961, Compound 23 | US106832...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  190nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50112244(CHEMBL3608680 | US10030025, Compound 5 | US1083676...)
Affinity DataKi:  219nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50112245(CHEMBL3608741 | US10030025, Compound 11 | US108367...)
Affinity DataKi:  244nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50341075((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)
Affinity DataKi:  250nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50112179(CHEMBL3608740 | US10030025, Compound 20 | US108367...)
Affinity DataKi:  573nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50112183(CHEMBL3608684 | US10214533, Compound 1 | US9969738...)
Affinity DataKi:  2.03E+3nMAssay Description:Binding affinity to rat NK3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50341076((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyb...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50341074((4-(2-methoxyphenyl)piperazin-1-yl)(3-phenyl-1H-py...)
Affinity DataKi:  1.20E+4nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed