TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Inhibition of rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Activity at rabbit bradykinin B1 receptor assessed by FLIPR assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Activity at rabbit bradykinin B1 receptor assessed by FLIPR assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Activity at rabbit bradykinin B1 receptor assessed by FLIPR assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 10.4nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 11.2nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 11.2nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 12.3nMAssay Description:Activity at rabbit bradykinin B1 receptor assessed by FLIPR assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonistic activity at rabbit bradykinin B1 receptor expressed in CHO-D cells assessed as effect on DAK-mediated calcium mobilizationMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 17.5nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 20.3nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 21.4nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 25.3nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 31.1nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 85.9nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 139nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >160nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 248nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 342nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 393nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 451nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 476nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.69E+3nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >4.00E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >4.00E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research And Development
Curated by ChEMBL
Affinity DataIC50: >6.47E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair