Compile Data Set for Download or QSAR
Report error Found 21 of ic50 for UniProtKB: P18090
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM25753(Artrenolol | 2-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataIC50: 5.30nMAssay Description:In vitro beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucose incorporation into glycog...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002132(CHEMBL38486 | (BRL 35,135)(4-{2-[2-(3-Chloro-pheny...)
Affinity DataIC50: 59nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272481(CHEMBL4128940)
Affinity DataIC50: 106nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272471(CHEMBL4127540)
Affinity DataIC50: 179nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272483(CHEMBL4128794)
Affinity DataIC50: 179nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002133((4-{2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-p...)
Affinity DataIC50: 190nMAssay Description:In vitro beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucose incorporation into glycog...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272482(CHEMBL4130151)
Affinity DataIC50: 426nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002132(CHEMBL38486 | (BRL 35,135)(4-{2-[2-(3-Chloro-pheny...)
Affinity DataIC50: 500nMAssay Description:In vitro beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucose incorporation into glycog...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataIC50: 600nMAssay Description:Compound was evaluated for its binding affinity towards beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272472(CHEMBL4128231)
Affinity DataIC50: 785nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50272473(CHEMBL4126588)
Affinity DataIC50: 1.42E+3nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002133((4-{2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-p...)
Affinity DataIC50: 3.30E+3nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002338(10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsul...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]DHA (Dihydroalprenolol) from beta-1 adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50019457(CHEMBL42084 | 2-Diethylamino-N-[4-(2-fluoro-benzoy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against beta-1 adrenergic receptor in rat brain using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50019968(CHEMBL143865 | 7-Ethyl-1,3,5-trimethyl-6,7-dihydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]DHA (Dihydroalprenolol) from beta-1 adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against beta-1 adrenergic receptor in rat brain using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50019458(CHEMBL45063 | N-[4-(2-Fluoro-benzoyl)-2,5-dimethyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against beta-1 adrenergic receptor in rat brain using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against beta-1 adrenergic receptor in rat brain using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002134(CL-316243 | CHEMBL32590 | 5-{2-[2-(3-Chloro-phenyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucose incorporation into glycog...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50002134(CL-316243 | CHEMBL32590 | 5-{2-[2-(3-Chloro-phenyl...)
Affinity DataIC50: 1.30E+6nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed