TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.100nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Negative allosteric modulation of alpha1 GABAA (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Binding affinity to GABA-A alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Binding affinity to GABA-A alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.700nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.730nMAssay Description:Binding affinity to GABA-A alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.794nMAssay Description:Binding affinity to GABBA alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Positive allosteric modulation of GABAA alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.830nMAssay Description:Binding affinity to GABA-A alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 0.880nMAssay Description:Binding affinity to GABA-A alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Positive allosteric modulation of GABAA alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 1.40nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Ligand Info
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2.40nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 2.60nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Clinic For Psychiatry
Curated by PDSP Ki Database
University Clinic For Psychiatry
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Electrophysiological experiments were performed on days 3 to 5 after the micro-injection of mRNA. During the experiment the oocytes were constantly s...More data for this Ligand-Target Pair