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TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataKd:  30nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  56nMAssay Description:Binding affinity to human HSP90B1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169936(CHEMBL3805415)
Affinity DataKd:  90nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  200nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50587146(CHEMBL5073759)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataKd:  220nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169939(CHEMBL3805519)
Affinity DataKd:  250nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50013895(CHEMBL3260480)
Affinity DataKd:  320nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169707(CHEMBL3805794)
Affinity DataKd:  350nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169714(CHEMBL3804936)
Affinity DataKd:  400nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50650754(CHEMBL5631777)
Affinity DataKd:  400nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50450701(CHEMBL4168274)
Affinity DataKd:  440nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM210959(4-(2-(2-hydroxybenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)...)
Affinity DataKd:  440nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169706(CHEMBL3804872)
Affinity DataKd:  440nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50650754(CHEMBL5631777)
Affinity DataKd:  460nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169708(CHEMBL3805768)
Affinity DataKd:  470nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50450704(CHEMBL560895 | SNX-2112)
Affinity DataKd:  484nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50649623(CHEMBL5619572)
Affinity DataKd:  520nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKd:  530nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169704(CHEMBL3805027)
Affinity DataKd:  550nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataKd:  620nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169705(CHEMBL3805428)
Affinity DataKd:  650nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169712(CHEMBL3805824)
Affinity DataKd:  670nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169710(CHEMBL3804875)
Affinity DataKd:  680nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169753(CHEMBL3805991)
Affinity DataKd:  720nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM210954(4-(2-(2-fluorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  720nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169843(CHEMBL3805286)
Affinity DataKd:  730nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169716(CHEMBL3805350)
Affinity DataKd:  750nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169713(CHEMBL3804981)
Affinity DataKd:  760nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169934(CHEMBL3805146)
Affinity DataKd:  810nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169784(CHEMBL3804944)
Affinity DataKd:  810nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50051099(CHEMBL3310671)
Affinity DataKd:  820nMAssay Description:Inhibition of recombinant Grp94 (unknown origin) assessed as tracer bound after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM210951(4-(2-(2-chlorobenzyl)-1H-pyrrol-1-yl)-2-(((1r,4r)-...)
Affinity DataKd:  830nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169711(CHEMBL3805965)
Affinity DataKd:  930nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169817(CHEMBL3805621)
Affinity DataKd:  960nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50051100(CHEMBL3310679)
Affinity DataKd:  1.08E+3nMAssay Description:Inhibition of recombinant Grp94 (unknown origin) assessed as tracer bound after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM210949(4-(2-benzyl-1H-pyrrol-1-yl)-2-(((1r,4r)-4-hydroxyc...)
Affinity DataKd:  1.13E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50087812(CHEMBL3426787)
Affinity DataKd:  1.14E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM210962(2-(((1r,4r)-4-hydroxycyclohexyl)amino)-4-(2-(2-met...)
Affinity DataKd:  1.15E+3nMpH: 7.3Assay Description:Assay buffer (25 μL, 20 mM HEPES at pH 7.3, 50 mM KCl, 5 mM MgCl2, 1 mM DTT, 20 mM Na2MoO4, 0.01% NP-40, and 0.5 mg mL−1 BGG) was added to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataKd:  1.20E+3nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169926(CHEMBL3805121)
Affinity DataKd:  1.30E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169878(CHEMBL3806252)
Affinity DataKd:  1.36E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50087812(CHEMBL3426787)
Affinity DataKd:  1.38E+3nMAssay Description:Binding affinity to recombinant GRP94 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169879(CHEMBL3805874)
Affinity DataKd:  1.39E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169875(CHEMBL3806136)
Affinity DataKd:  1.40E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169703(CHEMBL3805526)
Affinity DataKd:  1.50E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50051098(CHEMBL3310536)
Affinity DataKd:  1.50E+3nMAssay Description:Inhibition of recombinant Grp94 (unknown origin) assessed as tracer bound after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169941(CHEMBL3806120)
Affinity DataKd:  1.53E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
TargetEndoplasmin(Human)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50169877(CHEMBL3805920)
Affinity DataKd:  1.53E+3nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2017
Entry Details Article
PubMed
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