Compile Data Set for Download or QSAR
maximum 50k data
Found 174
LigandPNGBDBM50177232(4-(3-bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cycl...)
Affinity DataIC50:  5nMAssay Description:Anchorage-independent growth of transformed NIH3T3 cells in soft agarMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177232(4-(3-bromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cycl...)
Affinity DataIC50:  5.20nMAssay Description:Anchorage-independent growth of transformed NIH3T3 cells in soft agarMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079787(CHEMBL303859 | methyl 2-[1-[5-amino-2-isopropyl-6-...)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327974(CHEMBL1258797 | N-Benzyl,N-{2-[(4-Cyanophenyl)-(3-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327998(CHEMBL1258350 | N-(2-((4-cyano-2-fluorophenyl)((1-...)
Affinity DataIC50:  89nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327976(CHEMBL215476 | N-benzyl-N-(2-((4-cyanophenyl)((1-m...)
Affinity DataIC50:  90nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50065394((S)-2-(2-{[(S)-2-((R)-2-Amino-3-mercapto-propylami...)
Affinity DataIC50:  100nMAssay Description:Inhibition of post-translational processing of v-Ras protein in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13315(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50:  100nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327997(CHEMBL1258232 | N-(2-((4-cyanophenyl)((1-methyl-1H...)
Affinity DataIC50:  268nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327999(CHEMBL1258351 | N-(2-((5-cyanopyridin-2-yl)((1-met...)
Affinity DataIC50:  288nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13313(N-Benzyl-N-{2-[(4-cyanophenyl)-(3-methyl-3H-imidaz...)
Affinity DataIC50:  300nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327990(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50:  300nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079805(CHEMBL302834 | methyl 2-[1-[5-amino-6-sulfanyl-(5R...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059858((S)-2-((3Z,6E)-(2S,5S,8R)-8-Amino-2-benzyl-5-isopr...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327985(CHEMBL452319 | N-(2-((4-cyanophenyl)((1-methyl-1H-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327987(CHEMBL1257889 | N-(2-((4-cyanophenyl)((1-methyl-1H...)
Affinity DataIC50:  400nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059876(CHEMBL217423 | [(S)-1-[(S)-1-{(S)-2-Benzyloxy-1-[(...)
Affinity DataIC50:  420nMAssay Description:Inhibition of Ras-processing in H-Ras transformed NIH3T3 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079785(CHEMBL433102 | methyl 2-[1-[5-amino-6-sulfanyl-(E,...)
Affinity DataIC50:  490nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327975(CHEMBL215475 | N-benzyl-N-(2-((4-cyanophenyl)((1-m...)
Affinity DataIC50:  500nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50369376(CHEMBL1790751)
Affinity DataIC50:  500nMAssay Description:Inhibition of post-translational processing of v-Ras protein in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50059846(CHEMBL103575 | L-745631 | [(R)-4-((S)-2-Amino-3-me...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Ras processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327977(CHEMBL379511 | N-benzyl-N-(2-((4-cyanophenyl)((1-m...)
Affinity DataIC50:  600nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327984(CHEMBL1257647 | N-(2-((4-cyanophenyl)((1-methyl-1H...)
Affinity DataIC50:  650nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327986(CHEMBL1257770 | N-(2-((4-cyanophenyl)((1-methyl-1H...)
Affinity DataIC50:  800nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079790((S)-2-{[(2S,4S)-1-((E)-(2S,5R)-5-Amino-2-isopropyl...)
Affinity DataIC50:  840nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13311(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13314(5-Dimethylaminonaphthalene-1-sulfonic Acid Benzyl-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13308(N-benzyl-N-(2-{(4-bromophenyl)[(1-methyl-1H-imidaz...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13307(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-{2-[(...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50079800(CHEMBL303363 | methyl 2-[1-[5-amino-6-sulfanyl-(5R...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31423(ethylenediamine scaffold, 4)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50327991(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327993(1-methyl-1H-imidazole-4-sulfonic acid biphenyl-3-y...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079802(CHEMBL302025 | methyl 2-[1-[4-amino-5-sulfanyl-(E,...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079791(CHEMBL304823 | methyl 2-[1-[4-amino-5-sulfanyl-(E,...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079797(CHEMBL66788 | methyl 2-[1-[4-amino-5-sulfanyl-(E,4...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327994(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327983(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13316(1-Methyl-1H-imidazole-4-sulfonic Acid Biphenyl-4-y...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327992(1-methyl-1H-imidazole-4-sulfonic acid (3-cyanobenz...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097809((S)-2-[(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmet...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50403712(CHEMBL2092732)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibitory concentration against Farnesyltransferase for Farnesylation of H-ras protein InNIH 3T3 cells transformed with activated H-rasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327973(1-methyl-1H-imidazole-4-sulfonic acid benzyl-{2-[(...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327981(1-methyl-1H-imidazole-4-sulfonic acid (2-bromoally...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327978(CHEMBL1257299 | N-(2-((4-cyanophenyl)((1-methyl-1H...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327979(1-methyl-1H-imidazole-4-sulfonic acid allyl-{2-[(4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50327996(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of H-Ras farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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