Affinity DataKi: 0.100nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards human mu opioid receptor in CHO cells using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity towards human delta opioid receptor in CHO cells using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards mu opioid receptor in guinea pig brain membranes using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity towards human kappa opioid receptor in CHO cells using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Binding affinity towards kappa opioid receptor in guinea pig brain membranes using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Activity was evaluated in human delta opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activity was evaluated in human delta opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Activity was evaluated in human delta opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Activity was evaluated in human mu opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Activity was evaluated in human mu opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Activity was evaluated in human kappa opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Activity was evaluated in human kappa opioid receptors transfected with CHO cells by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair