Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50038006
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197693(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(6-methoxy-1,3...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197695(({[({[(2R,3S,4R,5R)-5-(5-fluoro-1,3-benzothiazol-2...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197694(({[({[(2R,3S,4R,5R)-5-(6-chloro-4-fluoro-1,3-benzo...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197696(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-[5-(trifluorom...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50195825(({[({[(2R,3S,4R,5R)-5-(7-fluoro-1-oxo-1,2-dihydroi...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197697(({[({[(2R,3S,4R,5R)-5-(1,3-benzothiazol-2-yl)-3,4-...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197696(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-[5-(trifluorom...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197698(({[({[(2R,3S,4R,5R)-5-(6-chloro-1,3-benzothiazol-2...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197696(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-[5-(trifluorom...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human cloned P2Y1 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197699(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-methoxy-1,3...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197694(({[({[(2R,3S,4R,5R)-5-(6-chloro-4-fluoro-1,3-benzo...)
Affinity DataEC50:  4.23E+3nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197700(({[({[(2R,3S,4R,5S)-3,4-dihydroxy-5-(1-methyl-1H-1...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197697(({[({[(2R,3S,4R,5R)-5-(1,3-benzothiazol-2-yl)-3,4-...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human cloned P2Y1 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197697(({[({[(2R,3S,4R,5R)-5-(1,3-benzothiazol-2-yl)-3,4-...)
Affinity DataEC50:  4.12E+3nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197701(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-1,3-...)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50: >2.00E+3nMAssay Description:Agonist activity at human cloned P2Y1 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Ucb-Group

Curated by ChEMBL
LigandPNGBDBM50197694(({[({[(2R,3S,4R,5R)-5-(6-chloro-4-fluoro-1,3-benzo...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human cloned P2Y1 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed