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Found 56 Enz. Inhib. hit(s) with all data for entry = 50018311
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated fo...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO3-AMC as substrate incubated fo...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421691(CHEMBL5275516)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO2-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421702(CHEMBL3236516)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human SENP1 catalytic domain assessed as reduction in deSUMOylation of RanGAP1-SUMO2 using RanGAP1-SUMO2 as substrate by fluorescence b...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human full-length recombinant SENP1More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human SENP1 catalytic domain assessed as reduction in deSUMOylation of RanGAP1-SUMO2 using RanGAP1-SUMO2 as substrate by fluorescence b...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM103827(SPI-02 | US11041859, Code SPI-02 | US9791447, Comp...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM50421692(CHEMBL5287963)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM103827(SPI-02 | US11041859, Code SPI-02 | US9791447, Comp...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421693(CHEMBL5269877)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421692(CHEMBL5287963)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421693(CHEMBL5269877)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM103828(SPI-03 | US11041859, Code SPI-03)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421702(CHEMBL3236516)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human full-length recombinant SENP1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421692(CHEMBL5287963)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103827(SPI-02 | US11041859, Code SPI-02 | US9791447, Comp...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM103826(SPI-01 | US11041859, Code SPI-01 | US9791447, Comp...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM50421693(CHEMBL5269877)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103826(SPI-01 | US11041859, Code SPI-01 | US9791447, Comp...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421699(CHEMBL5289490)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated fo...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591766(CHEMBL5188918)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM103828(SPI-03 | US11041859, Code SPI-03)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103830(SPI-05 | US11041859, Code SPI-05 | US9791447, Comp...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103831(SPI-06)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421698(CHEMBL5265789)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 3(Homo sapiens)TBA
LigandPNGBDBM103828(SPI-03 | US11041859, Code SPI-03)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of SENP3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421698(CHEMBL5265789)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50565347(CHEMBL4789677)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM103826(SPI-01 | US11041859, Code SPI-01 | US9791447, Comp...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421696(CHEMBL5278030)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421696(CHEMBL5278030)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421695(CHEMBL5281566)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421695(CHEMBL5281566)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421701(CHEMBL5287448)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM103830(SPI-05 | US11041859, Code SPI-05 | US9791447, Comp...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50355870(CHEMBL1910013)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of human SENP1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50565347(CHEMBL4789677)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421697(CHEMBL5277298)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 2(Homo sapiens (Human))TBA
LigandPNGBDBM50421694(CHEMBL5269942)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of SENP2 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM103830(SPI-05 | US11041859, Code SPI-05 | US9791447, Comp...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of SENP1 (unknown origin)More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50591762(CHEMBL470172)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of human SENP1 catalytic domain assessed as reduction in deSUMOylation of RanGAP1-SUMO2 using RanGAP1-SUMO2 as substrate by fluorescence b...More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50355868(CHEMBL1910011)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human SENP1More data for this Ligand-Target Pair
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TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421700(CHEMBL5289965)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421699(CHEMBL5289490)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO1-AMC as substrate incubated for 10 mins fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421701(CHEMBL5287448)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO2-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))TBA
LigandPNGBDBM50421701(CHEMBL5287448)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human recombinant His6 tagged SENP1 catalytic domain expressed in Escherichia coli BL21 (DE3) using SUMO3-AMC as substrate incubated fo...More data for this Ligand-Target Pair
In DepthDetails PubMed
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