Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50017774
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186292(2-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186309(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186269(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186270(2-benzyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tet...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186291(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186306(3-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186290(3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186278(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186311(3-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186297(CHEMBL209099 | N-isopropyl-7-(3-(piperidin-1-yl)pr...)
Affinity DataKi:  32.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186277(1-(7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoqui...)
Affinity DataKi:  36.7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186275(3-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2...)
Affinity DataKi:  38.1nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186285(CHEMBL208829 | N-isopropyl-7-(3-(piperidin-1-yl)pr...)
Affinity DataKi:  39.6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186300(1-(7-(3-(piperidin-1-yl)propoxy)-1,2,4,5-tetrahydr...)
Affinity DataKi:  48.8nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186295(2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2...)
Affinity DataKi:  70.1nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186288(2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  74.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed