Compile Data Set for Download or QSAR
maximum 50k data
Found 33
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM25524(17,18-dimethoxy-21-methyl-5,7-dioxa-21-azapentacyc...)
Affinity DataKi:  660nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50280897(CHEMBL281660 | Tetradecanoic acid (2S,3R)-2-(2-hyd...)
Affinity DataKi:  880nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50282658(((2R,3R)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-3-...)
Affinity DataKi:  1.47E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50280896(CHEMBL276429 | Tetradecanoic acid (2S,3R)-2-hydrox...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50282661(CHEMBL29762 | Tetradecanoic acid (2R,3S)-2-hydroxy...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86727(1-(5-isoquinolinesulfonyl)-2-methylpiperazine.2HCl...)
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM86729((R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cycloh...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50009723(2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...)
Affinity DataKi:  1.20E+4nMAssay Description:Effect of Phosphatidylserine on inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50282657(CHEMBL29668 | [(2S,3R)-2-(2-Hydroxy-ethyl)-5-oxo-t...)
Affinity DataKi:  1.86E+4nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50283971(CHEMBL153171 | Tetradecanoic acid (2S,3R)-2-hydrox...)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of [3H]-phorbol-12,13-dibutyrate from rat brain protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98660(US8497385, 18C)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98659(US8497385, 19B.0)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  2.85nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98661(US8497385, 19B.1)
Affinity DataIC50:  3.10nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98662(US8497385, 19B.2)
Affinity DataIC50:  3.80nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98663(US8497385, 19B.3)
Affinity DataIC50:  4.60nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM98664(US8497385, 19B.4)
Affinity DataIC50:  30nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92971(Amphiphile, VI)
Affinity DataIC50:  1.10E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92969(Amphiphile, IV)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92976(Amphiphile, XI)
Affinity DataIC50:  1.50E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50009723(2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...)
Affinity DataIC50:  1.90E+4nMAssay Description:Effect of PMA on inhibition of PKC alpha (Protein kinase C)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM50009723(2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...)
Affinity DataIC50:  1.90E+4nMAssay Description:Effect of PMA on inhibition of PKC alpha (Protein kinase C)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92978(Amphiphile, XIII)
Affinity DataIC50:  2.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92979(Amphiphile, XVI)
Affinity DataIC50:  2.60E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92980(Amphiphile, XVII)
Affinity DataIC50:  4.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92974(Amphiphile, IX)
Affinity DataIC50:  5.90E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92977(Amphiphile, XII)
Affinity DataIC50:  1.64E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92973(Amphiphile, VIII)
Affinity DataIC50:  1.91E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92972(Amphiphile, VII)
Affinity DataIC50:  2.46E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92968(Amphiphile, III)
Affinity DataIC50:  2.58E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92975(Amphiphile, X)
Affinity DataIC50:  4.08E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University

Curated by PDSP Ki Database
LigandPNGBDBM92970(Amphiphile, V)
Affinity DataIC50:  6.43E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed