Affinity DataEC50: 3.20nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 67nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 96nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 141nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 288nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 302nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at HCA3 receptor (unknown origin) expressed in CHOK1 cells assessed as ERK1/2 phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 331nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 692nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 724nMAssay Description:Agonist activity at human GPR109b expressed in human adipocytes assessed as decrease in intracellular cAMP level by HTRF assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 724nMAssay Description:Agonist activity at human GPR109b expressed in human adipocytes assessed as decrease in intracellular cAMP level by HTRF assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 851nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 891nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at human GPR109bMore data for this Ligand-Target Pair
Affinity DataEC50: 1.47E+3nMAssay Description:Activity at GPR109b assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.72E+3nMAssay Description:Activity at GPR109b assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.34E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.02E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.09E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.23E+3nMAssay Description:Agonist activity at human GPR109b expressed in human adipocytes assessed as decrease in intracellular cAMP level by HTRF assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.23E+3nMAssay Description:Agonist activity at human GPR109b expressed in human adipocytes assessed as decrease in intracellular cAMP level by HTRF assayChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.39E+3nMAssay Description:Agonistic activity at GPR109b by cAMP whole cell assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.98E+3nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+3nMAssay Description:Agonist activity at N-terminal HA-tagged GPR109b receptor transfected in forskolin-stimulated cells assessed as cAMP accumulation by flashplate assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 4.47E+3nMAssay Description:Agonist activity at GPR109b receptor transfected in CHOK1 cells assessed as inhibition of forskolin-induced cAMP generation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+3nMAssay Description:Activity at GPR109b in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair