Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 6841
TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153641BDBM153641(US8999982, Ref4)
Affinity DataIC50: 7.04E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153643BDBM153643(US8999982, Ref6)
Affinity DataIC50: 8.29E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153652BDBM153652(US8999982, 3-fluoro-4-((6-methoxy-7-(3- morpholino...)
Affinity DataIC50: 8.50E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153644BDBM153644(US8999982, Ref7)
Affinity DataIC50: 9.30E+3nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153648BDBM153648(US8999982, 3-chloro-4-((6,7- dimethoxyquinolin-4- ...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153649BDBM153649(US8999982, 5-((6,7-dimethoxyquinolin-4- yl)oxy)pyr...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153650BDBM153650(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153651BDBM153651(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-2-...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153645BDBM153645(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153646BDBM153646(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)ani...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153647BDBM153647(US8999982, 4-((6,7-dimethoxyquinolin-4- yl)oxy)-3-...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153640BDBM153640(US8999982, Ref3)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153642BDBM153642(US8999982, Ref5)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153653BDBM153653(US8999982, tert-butyl 4-(((4-(4-amino-2- fluorophe...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 50317324BDBM50317324(N-(4-(6,7-dimethoxyquinolin-4-yloxy)-3-fluoropheny...)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Lead Discovery Center

US Patent
LigandChemical structure of BindingDB Monomer ID 153639BDBM153639(US8999982, Ref2)
Affinity DataIC50: 1.00E+4nMpH: 8.0Assay Description:The principle behind this assay is based upon the binding and displacement of an Alexa Fluor 647-labeled tracer to the kinase of interest. Binding of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2015
Entry Details
US Patent