Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50011584
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi:  0.700nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076568(CHEMBL46542)
Affinity DataKi:  2.30nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076574(CHEMBL47240)
Affinity DataKi:  2.30nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi:  2.40nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50070096(CHEMBL298489)
Affinity DataKi:  9nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi:  15nMAssay Description:Binding affinity of the compound for gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  22nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi:  27nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076574(CHEMBL47240)
Affinity DataKi:  36nMAssay Description:Binding affinity for kappa opioid receptor by displacing [3H]U-69593 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  46nMAssay Description:Binding affinity of the compound for gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi:  49nMAssay Description:Binding affinity of the compound for gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076574(CHEMBL47240)
Affinity DataKi:  66nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi:  95nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076568(CHEMBL46542)
Affinity DataKi:  120nMAssay Description:Binding affinity for kappa opioid receptor by displacing [3H]U-69593 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi:  126nMAssay Description:Binding affinity for kappa opioid receptor by displacing [3H]U-69593 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi:  202nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi:  240nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  272nMAssay Description:Binding affinity of the compound for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  272nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi:  290nMAssay Description:Binding affinity of the compound for gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi:  330nMAssay Description:Binding affinity of the compound for gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi: >350nMAssay Description:Binding affinity for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi:  370nMAssay Description:Binding affinity for delta opioid receptor by displacing [3H]DADL was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi:  398nMAssay Description:Binding affinity of the compound for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  561nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi: >600nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50108346(CHEMBL295295 | Indole Derivative)
Affinity DataKi: >600nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi: >600nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi: >600nMAssay Description:Binding affinity of the compound for mu opioid receptor by displacing DAMGO was determined in [35S]-GTP gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi:  710nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi:  731nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding to p185erbB-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi: >750nMAssay Description:Binding affinity of the compound for gamma-S binding assay; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50070096(CHEMBL298489)
Affinity DataKi:  850nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding to p185erbB-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50076568(CHEMBL46542)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50070096(CHEMBL298489)
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108349(CHEMBL297839 | Indole Derivative)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108347(CHEMBL432117 | Indole Derivative)
Affinity DataKi: >4.30E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108348(CHEMBL296922 | Indole Derivative)
Affinity DataKi: >4.80E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50108351(CHEMBL45344 | Indole Derivative)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity for mu opioid receptor by displacing [3H]-DAMGO was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Niddk

Curated by ChEMBL
LigandPNGBDBM50451441(CHEMBL607396)
Affinity DataKi: >6.00E+3nMAssay Description:Binding affinity of the compound for kappa opioid receptor by displacing U-69,593 was determined in [35S]-GTP gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed