Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50015354
LigandPNGBDBM50155178((R)-2-Methyl-4-(4-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155156((R)-4-(6-Chloro-4-methyl-pyridazin-3-yl)-2-methyl-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155178((R)-2-Methyl-4-(4-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 15nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155158(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataIC50: 30nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155158(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 50nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155186((R)-2-Methyl-4-(4-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 58nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155156((R)-4-(6-Chloro-4-methyl-pyridazin-3-yl)-2-methyl-...)
Affinity DataIC50: 68nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155189(4-(6-Chloro-4-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155159((R)-4-(6-chloro-4-methylpyridazin-3-yl)-N-(6-fluor...)
Affinity DataIC50: 103nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155194(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 177nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155159((R)-4-(6-chloro-4-methylpyridazin-3-yl)-N-(6-fluor...)
Affinity DataIC50: 226nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155186((R)-2-Methyl-4-(4-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 251nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155181(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 279nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155189(4-(6-Chloro-4-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 301nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155182(4-Pyridazin-3-yl-piperazine-1-carboxylic acid (4-t...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155176(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155184(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155173((R)-4-(6-Chloro-5-methyl-pyridazin-3-yl)-2-methyl-...)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155163(4-(6-Chloro-4-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155180(4-(5-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 2.64E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155176(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 2.73E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155194(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 2.78E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155167(4-(6-Chloro-4-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155163(4-(6-Chloro-4-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 3.26E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155202(4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 3.83E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155203(4-(5-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 5.02E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155181(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 5.73E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155165(4-Pyridazin-3-yl-piperazine-1-carboxylic acid (4-i...)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155184(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 5.86E+3nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155160(4-(4-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 6.17E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155172((R)-4-(6-Chloro-5-methyl-pyridazin-3-yl)-2-methyl-...)
Affinity DataIC50: 8.12E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155179((R)-2-Methyl-4-(5-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 8.59E+3nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155190(4-(6-Phenyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155164(4-(6-Chloro-5-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155195(4-Phthalazin-1-yl-piperazine-1-carboxylic acid (4-...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155196(4-(6-Chloro-5-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155199(4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155162(4-(6-Phenyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155170(4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155174(4-Phthalazin-1-yl-piperazine-1-carboxylic acid (6-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155190(4-(6-Phenyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155164(4-(6-Chloro-5-methyl-pyridazin-3-yl)-piperazine-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155166(4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155191(4-(6-Methyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155174(4-Phthalazin-1-yl-piperazine-1-carboxylic acid (6-...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155170(4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155162(4-(6-Phenyl-pyridazin-3-yl)-piperazine-1-carboxyli...)
Affinity DataIC50: 1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50155187((R)-2-Methyl-4-(5-methyl-pyridazin-3-yl)-piperazin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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