Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50015861
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataKi:  0.510nMAssay Description:Inhibition of [3H]PGD-2 binding to human chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]PGD-2 binding to human chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]PGD-2 binding to human chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataIC50: 3nMAssay Description:Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PGD2-induced inositol phosphate formation at human chemoattractant receptor-homologous molecule expressed on TH2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]PGD-2 binding to human chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of beta-arrestin translocation at human Thromboxane A2 receptor in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of U-46,619-induced inositol phosphate accumulation at human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataIC50: 15nMAssay Description:Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataIC50: 26nMAssay Description:Inhibition of PGD2-induced inositol phosphate formation at human chemoattractant receptor-homologous molecule expressed on TH2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataIC50: 28nMAssay Description:Inhibition of beta-arrestin translocation at human chemoattractant receptor-homologous molecule expressed on TH2 cells in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataIC50: 29nMAssay Description:Inhibition of PGD2-induced inositol phosphate formation at human chemoattractant receptor-homologous molecule expressed on TH2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataKi:  540nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of U-46,619-induced inositol phosphate accumulation at human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of beta-arrestin translocation at human Thromboxane A2 receptor in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of beta-arrestin translocation at human Thromboxane A2 receptor in BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161747(3-{(R)-3-[(4-Fluoro-benzenesulfonyl)-methyl-amino]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PGD2-induced inositol phosphate formation at human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of beta-arrestin translocation at Thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161746(CHEMBL361812 | 3-[(R)-3-(4-Fluoro-benzenesulfonyla...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161748([3-((R)-4-Fluoro-benzenesulfonylamino)-1,2,3,4-tet...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]-PGD-2 binding to human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50161745({3-[((R)-4-Fluoro-benzenesulfonyl)-methyl-amino]-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PGD2-induced inositol phosphate formation at human Prostaglandin D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed