Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50016422
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168805(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  0.840nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168812(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  0.880nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168825(1-(3-Chloro-4-fluoro-phenyl)-3-[2-(3'-cyano-biphen...)
Affinity DataKi:  0.980nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168791(1-(3-Chloro-phenyl)-3-[2-(3'-cyano-biphenyl-4-yl)-...)
Affinity DataKi:  1.10nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168800(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168823(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  2.40nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168802(1-[2-(3'-Cyano-biphenyl-4-yl)-4-methylamino-butyl]...)
Affinity DataKi:  2.60nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168810(1-[2-(3'-Cyano-biphenyl-4-yl)-4-cyclopentylamino-b...)
Affinity DataKi:  3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168810(1-[2-(3'-Cyano-biphenyl-4-yl)-4-cyclopentylamino-b...)
Affinity DataKi:  3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168799(1-[2-(3'-Cyano-biphenyl-4-yl)-4-ethylamino-butyl]-...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168797(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  4.70nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168809(1-[2-(3'-Cyano-biphenyl-4-yl)-4-isopropylamino-but...)
Affinity DataKi:  5.60nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168814(1-[2-(3'-Cyano-biphenyl-4-yl)-4-dimethylamino-buty...)
Affinity DataKi:  7.40nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168804(1-(4-Chloro-phenyl)-3-[2-(3'-cyano-biphenyl-4-yl)-...)
Affinity DataKi:  9.20nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168821(1-[4-Cyclopentylamino-2-(3'-trifluoromethoxy-biphe...)
Affinity DataKi:  20nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168811(1-[4-Cyclopentylamino-2-(4-pyridin-3-yl-phenyl)-bu...)
Affinity DataKi:  24nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168792(1-[2-(3'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-...)
Affinity DataKi:  26nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168815(1-[4-Cyclopentylamino-2-(3'-fluoro-biphenyl-4-yl)-...)
Affinity DataKi:  37nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168824(1-[2-(4'-Cyano-biphenyl-4-yl)-4-cyclopentylamino-b...)
Affinity DataKi:  46nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168798(1-(2-Biphenyl-4-yl-4-cyclopentylamino-butyl)-3-(3,...)
Affinity DataKi:  50nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168817(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  100nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168801(1-[4-Cyclopentylamino-2-(4-pyridin-4-yl-phenyl)-bu...)
Affinity DataKi:  122nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168820(1-[2-(2'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-...)
Affinity DataKi:  130nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168793(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  135nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168816(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  205nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168819(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  240nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168803(1-[2-(4'-Chloro-biphenyl-4-yl)-4-cyclopentylamino-...)
Affinity DataKi:  280nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168808(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  300nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168822(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168795(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  1.22E+3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168796(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  1.64E+3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168818(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168807(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168794(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  1.85E+4nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50168806(1-[4-[1,4']Bipiperidinyl-1'-yl-2-(3,4-dichloro-phe...)
Affinity DataKi:  2.25E+4nMAssay Description:Inhibitory constant towards Human melanin-concentrating hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed