Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50016891
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174871(X1-Apc-DPhe-Arg-Trp-Z10-NH2 | CHEMBL372201)
Affinity DataEC50:  1nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174863(X3-Apc-DPhe-Arg-Trp-Z10-NH2 | CHEMBL411817)
Affinity DataEC50:  1nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174884(X1-Apc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL200276)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174078(Penta-Apc-DPhe-Arg-Trp-Gly-NH2 | 1-Pentanoylamino-...)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174882(X2-Apc-DPhe-Arg-Trp-Z8-NH2 | CHEMBL425992)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174869(X3-Apc-DPhe-Arg-Trp-Z8-NH2 | CHEMBL409588)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174867(X3-Apc-DPhe-Arg-Trp-Z2-NH2 | CHEMBL372200)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174866(X1-Apc-DPhe-Arg-Trp-Z8-NH2 | CHEMBL444880)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174879(X2-Apc-DPhe-Arg-Trp-Z4-NH2 | CHEMBL370665)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174864(X2-Apc-DPhe-Arg-Trp-Z3-NH2 | CHEMBL200614)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174878(X2-Apc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL373259)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174889(X2-Apc-DPhe-Arg-Trp-Z2-NH2 | CHEMBL434186)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174883(X3-Apc-DPhe-Arg-Trp-Z3-NH2 | CHEMBL196773)
Affinity DataEC50:  3nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174868(X3-Apc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL409589)
Affinity DataEC50:  3nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174876(X1-Apc-DPhe-Arg-Trp-Z3-NH2 | CHEMBL383143)
Affinity DataEC50:  3nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174873(X1-Apc-DPhe-Arg-Trp-Z4-NH2 | CHEMBL373016)
Affinity DataEC50:  5nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174862(X3-Apc-DPhe-Arg-Trp-Z4-NH2 | CHEMBL372829)
Affinity DataEC50:  5nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50121885((S)-2-{(R)-2-[(S)-2-Butyrylamino-3-(3H-imidazol-4-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity in HEK293 cells transfected with human MC1R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174886(X3-5-BrAtc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL381007)
Affinity DataEC50:  11nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174874(Bu-His-DPhe-Arg-2-Nal-Gly-NH2 | CHEMBL369867)
Affinity DataEC50:  14nMAssay Description:Agonist activity in HEK293 cells transfected with human MC1R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174870(X1-5-BrAtc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL382930)
Affinity DataEC50:  15nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174875(X2-5-BrAtc-DPhe-Arg-Trp-Z9-NH2 | CHEMBL414670)
Affinity DataEC50:  15nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50121885((S)-2-{(R)-2-[(S)-2-Butyrylamino-3-(3H-imidazol-4-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174874(Bu-His-DPhe-Arg-2-Nal-Gly-NH2 | CHEMBL369867)
Affinity DataEC50:  25nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50121884(Penta-5-BrAtc-DPhe-Arg-Trp-Gly-NH2 | 5-Bromo-2-pen...)
Affinity DataEC50:  35nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174872(Bu-Apc-DPhe-Arg-2-Nal-Z9-NH2 | CHEMBL200668)
Affinity DataEC50:  39nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174881(Bu-Apc-DPhe-Arg-2-Nal-Z2-NH2 | CHEMBL372789)
Affinity DataEC50:  44nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174880(Penta-Apc-DPhe-Arg-2-Nal-Gly-NH2 | CHEMBL199740)
Affinity DataEC50:  50nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174885(Bu-5BrAtc-DPhe-Arg-2-Nal-Z9-NH2 | CHEMBL200449)
Affinity DataEC50:  72nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174888(Bu-Apc-DPhe-Arg-2-Nal-Z10-NH2 | CHEMBL382273)
Affinity DataEC50:  85nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174890(Bu-Apc-DPhe-Arg-2-Nal-Z4-NH2 | CHEMBL436296)
Affinity DataEC50:  90nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174887(Bu-Apc-DPhe-Arg-2-Nal-Z8-NH2 | CHEMBL200270)
Affinity DataEC50:  110nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174075(Penta-Apc-DPhe-Arg-Trp-NH2 | 1-Pentanoylamino-4-ph...)
Affinity DataEC50:  130nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174865(Penta-5-BrAtc-DPhe-Arg-2-Nal-Gly-NH2 | CHEMBL37121...)
Affinity DataEC50:  200nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174877(Bu-Apc-DPhe-Arg-2-Nal-Z3-NH2 | CHEMBL369915)
Affinity DataEC50:  220nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174075(Penta-Apc-DPhe-Arg-Trp-NH2 | 1-Pentanoylamino-4-ph...)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity in HEK293 cells transfected with human MC1R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174865(Penta-5-BrAtc-DPhe-Arg-2-Nal-Gly-NH2 | CHEMBL37121...)
Affinity DataEC50:  2.90E+3nMAssay Description:Agonist activity in HEK293 cells transfected with human MC1R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed