Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50016964
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175811BDBM50175811(N-(4-{[4-(1H-benzoimidazol-2-yl)phenylamino]methyl...)
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175813BDBM50175813(N-(4-{[5-(1H-benzoimidazol-2-yl)-pyridin-2-ylamino...)
Affinity DataIC50: 290nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175823BDBM50175823(N-{4-[4-(1H-benzoimidazol-2-yl)-phenylcarbamoyl]-p...)
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175822BDBM50175822(1-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-(3-bromo-...)
Affinity DataIC50: 930nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175821BDBM50175821(N-(4-((4-(1H-imidazo[4,5-c]pyridin-2-yl)phenylamin...)
Affinity DataIC50: 930nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175803BDBM50175803(3-bromo-N-(4-(5,6-dimethyl-1H-benzo[d]imidazol-2-y...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175819BDBM50175819(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-bromo-4-e...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175807BDBM50175807(3-bromo-N-(4-(4,5-dimethyl-1H-benzo[d]imidazol-2-y...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175825BDBM50175825(3-bromo-4-ethoxy-N-(4-(5-methyl-1H-benzo[d]imidazo...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175810BDBM50175810(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-bromo-4-p...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175824BDBM50175824(3-bromo-4-ethoxy-N-(4-(4-methyl-1H-benzo[d]imidazo...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175806BDBM50175806(3-bromo-N-(4-(4,7-dimethyl-1H-benzo[d]imidazol-2-y...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175812BDBM50175812(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-bromo-4-m...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175815BDBM50175815(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-4-methoxy-3...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175805BDBM50175805(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-(1H-indaz...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175816BDBM50175816(4'-hydroxy-6-methoxy-biphenyl-3-carboxylic acid [4...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175818BDBM50175818(4-(1H-benzo[d]imidazol-2-yl)-N-(3-bromo-4-methoxyp...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175817BDBM50175817(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-bromo-4-m...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175820BDBM50175820(N-(3-bromo-4-methoxybenzyl)-4-(1H-benzo[d]imidazol...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175809BDBM50175809(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-2-(3-bromo-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175804BDBM50175804(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-chloro-4-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175814BDBM50175814(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-fluoro-4-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175808BDBM50175808(N-(4-(1H-benzo[d]imidazol-2-yl)phenyl)-3-bromo-4-m...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against heparanase from human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed