Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 2386
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 10nM EC50:  0.590nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 11nM EC50:  0.840nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19953(5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dihydroquina...)
Affinity DataIC50: 47nM EC50:  13nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19962(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromene-4-th...)
Affinity DataIC50: 1.34E+3nM EC50:  14nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19954(3-(3-fluoro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 102nM EC50:  20nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19951(7-hydroxy-5-(hydroxymethyl)-3-(4-hydroxyphenyl)-3,...)
Affinity DataIC50: 24nM EC50:  4.46E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM17289(folliculin | (1S,10R,11S,15S)-5-hydroxy-15-methylt...)
Affinity DataIC50: 31nM EC50:  26nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM17289(folliculin | (1S,10R,11S,15S)-5-hydroxy-15-methylt...)
Affinity DataIC50: 29nM EC50:  166nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19957(5-ethyl-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydroq...)
Affinity DataIC50: 156nM EC50:  53nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 61nM EC50:  73nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19947(5-ethyl-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydroq...)
Affinity DataIC50: 265nM EC50:  62nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19910(5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dihydroquina...)
Affinity DataIC50: 179nM EC50:  76nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19956(7-hydroxy-3-(4-hydroxyphenyl)-5-methyl-3,4-dihydro...)
Affinity DataIC50: 79nM EC50:  222nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19912(5,7-dihydroxy-3-(4-hydroxy-2-methylphenyl)-3,4-dih...)
Affinity DataIC50: 422nM EC50:  111nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19914(3-(3-fluoro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 650nM EC50:  117nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19951(7-hydroxy-5-(hydroxymethyl)-3-(4-hydroxyphenyl)-3,...)
Affinity DataIC50: 121nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19943(7-hydroxy-3-(4-hydroxyphenyl)-5-methyl-3,4-dihydro...)
Affinity DataIC50: 317nM EC50:  136nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19955(5,7-dihydroxy-3-(4-hydroxy-3-methylphenyl)-3,4-dih...)
Affinity DataIC50: 658nM EC50:  160nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19958(5,7-dihydroxy-3-(5-hydroxypyridin-2-yl)-3,4-dihydr...)
Affinity DataIC50: 515nM EC50:  173nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19933(2-butyl-5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dihy...)
Affinity DataIC50: 178nMpH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19915(3-(2-fluoro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 256nM EC50:  190nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19933(2-butyl-5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dihy...)
Affinity DataIC50: 249nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19916(3-(2-chloro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 263nM EC50:  251nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19920(5,7-dihydroxy-3-(5-hydroxypyridin-2-yl)-3,4-dihydr...)
Affinity DataIC50: 3.53E+3nM EC50:  358nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19922(5,7-dihydroxy-3-(4-hydroxyphenyl)-8-iodo-3,4-dihyd...)
Affinity DataIC50: 4.08E+3nM EC50:  593nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19952(7-hydroxy-3-(4-hydroxyphenyl)-5-(prop-1-en-2-yl)-3...)
Affinity DataIC50: 2.30E+3nM EC50:  729nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19948(5-ethenyl-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydr...)
Affinity DataIC50: 1.70E+4nM EC50:  750nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19954(3-(3-fluoro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 3.08E+3nM EC50:  776nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19928(5,7-dihydroxy-3-(3-hydroxyphenyl)-3,4-dihydroquina...)
Affinity DataIC50: 3.84E+3nM EC50:  904nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 1.97E+3nM EC50:  956nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19927(7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydroquinazoli...)
Affinity DataIC50: 8.61E+3nM EC50:  961nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19936(5,7-dihydroxy-3-(4-hydroxyphenyl)-2-sulfanyl-3,4-d...)
Affinity DataIC50: 1.11E+4nM EC50:  983nMpH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19962(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromene-4-th...)
Affinity DataIC50: 5.59E+4nM EC50:  1.13E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19915(3-(2-fluoro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 7.49E+3nM EC50:  1.14E+3nMpH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19913(3-(3-chloro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 7.21E+3nM EC50:  1.18E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19917(5,7-dihydroxy-3-(4-hydroxy-3-methylphenyl)-3,4-dih...)
Affinity DataIC50: 7.49E+3nM EC50:  1.25E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19931(2-ethyl-5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dihy...)
Affinity DataIC50: 5.75E+3nM EC50:  1.26E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19924(5,7-dihydroxy-3-(4-hydroxyphenyl)-8-methyl-3,4-dih...)
Affinity DataIC50: 1.28E+3nM EC50:  8.87E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19938(2,5,7-trihydroxy-3-(4-hydroxyphenyl)-3,4-dihydroqu...)
Affinity DataIC50: 9.38E+3nM EC50:  1.31E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19916(3-(2-chloro-4-hydroxyphenyl)-5,7-dihydroxy-3,4-dih...)
Affinity DataIC50: 6.25E+3nM EC50:  1.43E+3nMpH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19957(5-ethyl-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydroq...)
Affinity DataIC50: 2.26E+3nM EC50:  1.46E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19930(5,7-dihydroxy-3-(4-hydroxyphenyl)-2-methyl-3,4-dih...)
Affinity DataIC50: 1.14E+4nM EC50:  1.58E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19925(5,7-dihydroxy-3-(4-hydroxyphenyl)-6-iodo-3,4-dihyd...)
Affinity DataIC50: 3.97E+3nM EC50:  1.64E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19956(7-hydroxy-3-(4-hydroxyphenyl)-5-methyl-3,4-dihydro...)
Affinity DataIC50: 1.75E+3nM EC50:  1.67E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19929(5,7-dihydroxy-3-phenyl-3,4-dihydroquinazolin-4-one...)
Affinity DataIC50: 1.85E+4nM EC50:  1.72E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19923(5,7-dihydroxy-3-(4-hydroxyphenyl)-6,8-diiodo-3,4-d...)
Affinity DataIC50: 1.23E+4nM EC50:  1.97E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19936(5,7-dihydroxy-3-(4-hydroxyphenyl)-2-sulfanyl-3,4-d...)
Affinity DataIC50: 6.99E+3nM EC50:  1.99E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Bristol-Myers Squibb

LigandPNGBDBM19942(5-amino-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydroq...)
Affinity DataIC50: 8.24E+3nM EC50:  2.06E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19943(7-hydroxy-3-(4-hydroxyphenyl)-5-methyl-3,4-dihydro...)
Affinity DataIC50: 9.64E+3nM EC50:  2.39E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Bristol-Myers Squibb

LigandPNGBDBM19955(5,7-dihydroxy-3-(4-hydroxy-3-methylphenyl)-3,4-dih...)
Affinity DataIC50: 2.85E+3nM EC50:  2.41E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2008
Entry Details Article
PubMed
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