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Found 19 Enz. Inhib. hit(s) with all data for entry = 50041464
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002726(CHEMBL2371933)
Affinity DataKi:  0.910nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002718(CHEMBL385281)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002725(CHEMBL374468)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002728(CHEMBL218825)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002723(CHEMBL265166)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002717(CHEMBL216712)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002727(CHEMBL266651)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002716(CHEMBL383996)
Affinity DataKi:  9.10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002719(CHEMBL412179)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002715(CHEMBL376223)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002720(CHEMBL219356)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002724(CHEMBL428990)
Affinity DataKi:  74nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002722(CHEMBL415851)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002713(CHEMBL425467)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002698(CHEMBL437110)
Affinity DataKi:  263nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50411186(CHEMBL218698)
Affinity DataKi:  407nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002721(CHEMBL415850)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002714(CHEMBL216716)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed