Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 2672
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23229([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 390nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
University of Mississippi

LigandPNGBDBM60537(US9115061, XVII)
Affinity DataIC50: 390nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23229([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 1.75E+3nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 2.03E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 2.64E+3nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23229([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 2.66E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23227([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 2.72E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 2.80E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23227([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 3.13E+3nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23227([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 4.88E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 5.80E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23228([(2-cyano-4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)me...)
Affinity DataIC50: 5.91E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23229([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 6.31E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23227([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 6.76E+3nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23228([(2-cyano-4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)me...)
Affinity DataIC50: 8.25E+3nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 9.54E+3nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23228([(2-cyano-4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)me...)
Affinity DataIC50: 1.09E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23229([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 1.14E+4nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23231(7-{2-[3-cyano-4-(formamidoformic acid)phenyl]ethox...)
Affinity DataIC50: 1.36E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23231(7-{2-[3-cyano-4-(formamidoformic acid)phenyl]ethox...)
Affinity DataIC50: 1.71E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23224(7-{[4-(formamidoformic acid)-3-methoxyphenyl]metho...)
Affinity DataIC50: 4.83E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23224(7-{[4-(formamidoformic acid)-3-methoxyphenyl]metho...)
Affinity DataIC50: 6.40E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23228([(2-cyano-4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)me...)
Affinity DataIC50: 8.69E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23224(7-{[4-(formamidoformic acid)-3-methoxyphenyl]metho...)
Affinity DataIC50: 8.73E+4nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataIC50: 9.25E+4nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23225(7-{2-[4-(formamidoformic acid)phenyl]ethoxy}-5-hyd...)
Affinity DataIC50: 9.67E+4nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataIC50: 1.23E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23228([(2-cyano-4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)me...)
Affinity DataIC50: 1.79E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23227([(4-{2-[(5-hydroxy-2-{[(4-methoxyphenyl)methyl]car...)
Affinity DataIC50: 1.87E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23226(7-{2-[4-(formamidoformic acid)-3-methoxyphenyl]eth...)
Affinity DataIC50: 1.91E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23226(7-{2-[4-(formamidoformic acid)-3-methoxyphenyl]eth...)
Affinity DataIC50: 2.25E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23226(7-{2-[4-(formamidoformic acid)-3-methoxyphenyl]eth...)
Affinity DataIC50: 2.25E+5nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23226(7-{2-[4-(formamidoformic acid)-3-methoxyphenyl]eth...)
Affinity DataIC50: 2.25E+5nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23224(7-{[4-(formamidoformic acid)-3-methoxyphenyl]metho...)
Affinity DataIC50: 2.32E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23224(7-{[4-(formamidoformic acid)-3-methoxyphenyl]metho...)
Affinity DataIC50: 2.32E+5nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Bovine)
University of Mississippi

LigandPNGBDBM23225(7-{2-[4-(formamidoformic acid)phenyl]ethoxy}-5-hyd...)
Affinity DataIC50: 2.41E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23225(7-{2-[4-(formamidoformic acid)phenyl]ethoxy}-5-hyd...)
Affinity DataIC50: 2.41E+5nMpH: 7.0 T: 2°CAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23225(7-{2-[4-(formamidoformic acid)phenyl]ethoxy}-5-hyd...)
Affinity DataIC50: 2.41E+5nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetL-lactate dehydrogenase(malaria parasite P. falciparum)
University of Mississippi

LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataIC50: 2.00E+6nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, cytoplasmic(Pig)
University of Mississippi

LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataIC50: 2.00E+6nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Pig)
University of Mississippi

LigandPNGBDBM23222(carbamoylformic acid | Oxalamic acid | Oxamidic Ac...)
Affinity DataIC50: 2.00E+6nMAssay Description:LDH was assayed spectrophotometrically for reduction of pyruvate using NADH by recording the changed in absorbance at 340 nm. The reaction was initia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2008
Entry Details Article
PubMed