Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50033459
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099348BDBM50099348(2-(2,4-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099358BDBM50099358(2-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099373BDBM50099373(2-(4-Ethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piper...)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099345BDBM50099345(2-(2,5-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099343BDBM50099343(2-(2-Fluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 13nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099367BDBM50099367(4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099342BDBM50099342(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099349BDBM50099349(2-(2,3-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099374BDBM50099374(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099352BDBM50099352(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099341BDBM50099341(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099347BDBM50099347(2-(3,4-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 22nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099338BDBM50099338(2-(Benzo[1,3]dioxol-5-yloxy)-4-[5-(4-fluoro-phenyl...)
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099334BDBM50099334(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 25nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099353BDBM50099353(2-(2,6-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 34.3nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099365BDBM50099365(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099333BDBM50099333(2-(3,5-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099329BDBM50099329(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 56nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099328BDBM50099328(2-(Biphenyl-4-yloxy)-4-[5-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 60nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099364BDBM50099364(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 75nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099340BDBM50099340(2-(4-tert-Butyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 79nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099360BDBM50099360(4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 82nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345778BDBM50345778(ethyl 4-(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-...)
Affinity DataIC50: 85.4nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099350BDBM50099350(4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 89.7nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099346BDBM50099346(2-(3-Fluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 95nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099366BDBM50099366(2-(4-Chloro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 114nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099332BDBM50099332((4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imi...)
Affinity DataIC50: 119nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099359BDBM50099359(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 130nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099335BDBM50099335(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 132nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345779BDBM50345779(2-(2-(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-...)
Affinity DataIC50: 134nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345780BDBM50345780(3-(2-(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-...)
Affinity DataIC50: 151nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099357BDBM50099357(2-(3,4-Dichloro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataIC50: 165nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099356BDBM50099356(4-(4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-i...)
Affinity DataIC50: 174nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099337BDBM50099337(4-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 177nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099371BDBM50099371(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 191nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345781BDBM50345781(2-(3,4-difluorophenoxy)-4-(4-(4-fluorophenyl)-1-(p...)
Affinity DataIC50: 209nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099351BDBM50099351(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 215nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099362BDBM50099362(2-(4-Fluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-pipe...)
Affinity DataIC50: 300nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099372BDBM50099372(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 312nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345782BDBM50345782(4-(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imi...)
Affinity DataIC50: 317nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099354BDBM50099354(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 406nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345783BDBM50345783(2-(3-(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-...)
Affinity DataIC50: 453nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099361BDBM50099361(3-{4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imid...)
Affinity DataIC50: 599nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
University College of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099336BDBM50099336(4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazo...)
Affinity DataIC50: 650nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed