Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50030408
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM94597((Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295708(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295714(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295718(6-(3-(4-(3,4-dichlorophenoxy)piperidin-1-yl)propyl...)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295710(10-(4-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295715(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295709(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295720(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295723(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295717(10-((1-(3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahyd...)
Affinity DataIC50: 46nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295716(10-((1-(3-((1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295718(6-(3-(4-(3,4-dichlorophenoxy)piperidin-1-yl)propyl...)
Affinity DataIC50: 58nMAssay Description:Inhibition of histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295726(3-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 69nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295725(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 72nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM22874(CHEMBL914 | Allegra | 2-(4-{1-hydroxy-4-[4-(hydrox...)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM22874(CHEMBL914 | Allegra | 2-(4-{1-hydroxy-4-[4-(hydrox...)
Affinity DataIC50: 78nMAssay Description:Inhibition of histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295722(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 88nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295727(3-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 105nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295724(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 123nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295711(10-(2-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 124nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295721(3-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 323nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295712(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295713(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydr...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Phrama.

Curated by ChEMBL
LigandPNGBDBM50295719(5-chloro-2-(1-(3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-t...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed