Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50031261
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310094((7-carbamoyl-8H-indeno[1,2-d]thiazol-4-yloxy)methy...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310095((7-(methylcarbamoyl)-8H-indeno[1,2-d]thiazol-4-ylo...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310093((7-(pyrimidin-5-yl)-8H-indeno[1,2-d]thiazol-4-ylox...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310086((7-chloro-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310083((7-methyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310091((7-(pyridin-3-yl)-8H-indeno[1,2-d]thiazol-4-yloxy)...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310092((7-(pyridin-4-yl)-8H-indeno[1,2-d]thiazol-4-yloxy)...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310088((6,7-difluoro-8H-indeno[1,2-d]thiazol-4-yloxy)meth...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50293594(5-(2-amino-5-isobutylthiazol-4-yl)furan-2-ylphosph...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310087((6,7-dimethyl-8H-indeno[1,2-d]thiazol-4-yloxy)meth...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310084((7-ethyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylpho...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310082((8H-indeno[1,2-d]thiazol-4-yloxy)methylphosphonic ...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310085((7-fluoro-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310089((7-phenyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310090((7-(pyridin-2-yl)-8H-indeno[1,2-d]thiazol-4-yloxy)...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50302500((2-amino-8H-indeno[1,2-d]thiazol-4-yloxy)methylpho...)
Affinity DataIC50:  124nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310081((2-bromo-8H-indeno[1,2-d]thiazol-4-yloxy)methylpho...)
Affinity DataIC50:  772nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310080((2-chloro-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  908nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50310079((2-methyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50:  995nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed