Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50039016
Target5-hydroxytryptamine receptor 6(Mouse)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86428BDBM86428(SB-258585)
Affinity DataKi:  0.75nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304001BDBM50304001([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Mouse)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304001BDBM50304001([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304003BDBM50304003(1-Naphthyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)m...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304003BDBM50304003(1-Naphthyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)m...)
Affinity DataKi:  15nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303997BDBM50303997(2-Benzyl-4-(4-methylpiperazin-1-yl)-1H-benzimidazo...)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304002BDBM50304002(2-(1-Naphthylmethyl)-4-piperazin-1-yl-1H-benzimida...)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304002BDBM50304002(2-(1-Naphthylmethyl)-4-piperazin-1-yl-1H-benzimida...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303999BDBM50303999(4-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H...)
Affinity DataKi:  17nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304000BDBM50304000(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Affinity DataKi:  27nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303998BDBM50303998(2-Benzyl-4-piperazin-1-yl-1H-benzimidazole | CHEMB...)
Affinity DataKi:  31nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of serotonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304001BDBM50304001([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304000BDBM50304000(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Affinity DataKi:  36.2nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303999BDBM50303999(4-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303998BDBM50303998(2-Benzyl-4-piperazin-1-yl-1H-benzimidazole | CHEMB...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303997BDBM50303997(2-Benzyl-4-(4-methylpiperazin-1-yl)-1H-benzimidazo...)
Affinity DataKi:  66.8nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303996BDBM50303996(Phenyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)metha...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304006BDBM50304006(5-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304005BDBM50304005(2-(2-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimida...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304004BDBM50304004(5-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303990BDBM50303990(2-Naphthyl-(5-piperazin-1-yl-1H-benzimidazol-2-yl)...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303991BDBM50303991([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303992BDBM50303992([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303993BDBM50303993([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303994BDBM50303994([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304001BDBM50304001([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304003BDBM50304003(1-Naphthyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)m...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303995BDBM50303995([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304007BDBM50304007(2-(1-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimida...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303988BDBM50303988(2-Benzyl-5-(4-methylpiperazin-1-yl)-1H-benzimidazo...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303989BDBM50303989(2-Benzyl-5-piperazin-1-yl-1H-benzimidazole | CHEMB...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303999BDBM50303999(4-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304000BDBM50304000(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304002BDBM50304002(2-(1-Naphthylmethyl)-4-piperazin-1-yl-1H-benzimida...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303997BDBM50303997(2-Benzyl-4-(4-methylpiperazin-1-yl)-1H-benzimidazo...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303998BDBM50303998(2-Benzyl-4-piperazin-1-yl-1H-benzimidazole | CHEMB...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304004BDBM50304004(5-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304005BDBM50304005(2-(2-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimida...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304006BDBM50304006(5-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303995BDBM50303995([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303996BDBM50303996(Phenyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)metha...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080167BDBM50080167(4-(4-methylpiperazin-1-yl)-1H-benzimidazole | 4-(4...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303988BDBM50303988(2-Benzyl-5-(4-methylpiperazin-1-yl)-1H-benzimidazo...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303989BDBM50303989(2-Benzyl-5-piperazin-1-yl-1H-benzimidazole | CHEMB...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303990BDBM50303990(2-Naphthyl-(5-piperazin-1-yl-1H-benzimidazol-2-yl)...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303991BDBM50303991([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303992BDBM50303992([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303993BDBM50303993([5-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50303994BDBM50303994([4-(4-Methylpiperazin-1-yl)-1H-benzimidazol-2-yl](...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304007BDBM50304007(2-(1-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimida...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed