Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50041780
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415407(CHEMBL612138)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415421(CHEMBL603112)
Affinity DataEC50:  3.98nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415424(CHEMBL601638)
Affinity DataEC50:  3.98nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415399(CHEMBL601440)
Affinity DataEC50:  7.94nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415425(CHEMBL605367)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415423(CHEMBL601637)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415428(CHEMBL604131)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415384(CHEMBL590495)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415401(CHEMBL601441)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415402(CHEMBL600821)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415403(CHEMBL604537)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415372(CHEMBL600827)
Affinity DataEC50:  15.8nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415412(CHEMBL601882)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415385(CHEMBL598743)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415422(CHEMBL603921)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415391(CHEMBL599328)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415416(CHEMBL600833)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414954(CHEMBL575966)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415409(CHEMBL604543)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415417(CHEMBL600834)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415429(CHEMBL601428)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415380(CHEMBL600020)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415406(CHEMBL603500)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414955(CHEMBL576138)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415404(CHEMBL602892)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415382(CHEMBL590982)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415373(CHEMBL600421)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415376(CHEMBL600629)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415398(CHEMBL601233)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415381(CHEMBL600021)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415410(CHEMBL602691)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414954(CHEMBL575966)
Affinity DataIC50: 316nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415418(CHEMBL608867)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415392(CHEMBL599347)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415393(CHEMBL605356)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415379(CHEMBL604751)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415374(CHEMBL605986)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415400(CHEMBL591455)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415369(CHEMBL601449)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415413(CHEMBL591927)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415371(CHEMBL590739)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415368(CHEMBL604752)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415414(CHEMBL601670)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415426(CHEMBL592645)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415405(CHEMBL603096)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415387(CHEMBL599126)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415411(CHEMBL603706)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414954(CHEMBL575966)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415420(CHEMBL592158)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415389(CHEMBL599127)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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