Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50032200
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325913(2-(3-(2-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  15nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325914(2-(3-(3-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  33nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325924(2-((3-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  50nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325908(2-(3-phenoxypropoxy)pyrido[2,3-d]pyrimidin-4(3H)-o...)
Affinity DataIC50:  130nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325920(2-((2-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  220nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325921(2-((3-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  230nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325915(2-(3-(4-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  230nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325910(2-(3-(2-fluorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  250nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325911(2-(3-(3-fluorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  370nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325907(2-(cinnamyloxy)pyrido[2,3-d]pyrimidin-4(3H)-one | ...)
Affinity DataIC50:  370nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50:  400nMAssay Description:Displacement of radioligand from rat GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325927(2-(2-m-Tolyl-ethoxymethyl)-3H-pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  410nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325926(2-(2-o-Tolyl-ethoxymethyl)-3H-pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  440nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325916(2-(3-(o-tolyloxy)propoxy)pyrido[2,3-d]pyrimidin-4(...)
Affinity DataIC50:  450nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325923(2-((2-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  600nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325922(2-((4-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  630nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325924(2-((3-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  640nMAssay Description:Displacement of radioligand from rat GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325900(2-((phenethyloxy)methyl)pyrido[2,3-d]pyrimidin-4(3...)
Affinity DataIC50:  670nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325896(2-(4-phenylbutoxy)pyrido[2,3-d]pyrimidin-4(3H)-one...)
Affinity DataIC50:  840nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325917(2-(3-(m-tolyloxy)propoxy)pyrido[2,3-d]pyrimidin-4(...)
Affinity DataIC50:  860nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325909(CHEMBL1223958 | N-((3,4-dihydro-4-oxopyrido[2,3-d]...)
Affinity DataIC50:  920nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325912(2-(3-(4-fluorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325925(2-((4-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325913(2-(3-(2-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of radioligand from rat GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325930(2-((3-methoxyphenethyloxy)methyl)pyrido[2,3-d]pyri...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325929(2-((2-methoxyphenethyloxy)methyl)pyrido[2,3-d]pyri...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325922(2-((4-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50:  2.70E+3nMAssay Description:Displacement of radioligand from rat GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325928(2-(2-p-Tolyl-ethoxymethyl)-3H-pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  4.30E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325931(2-((4-methoxyphenethyloxy)methyl)pyrido[2,3-d]pyri...)
Affinity DataIC50:  4.40E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325904(2-(4-phenylbutyl)pyrido[2,3-d]pyrimidin-4(3H)-one ...)
Affinity DataIC50:  4.40E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325918(2-(3-(p-tolyloxy)propoxy)pyrido[2,3-d]pyrimidin-4(...)
Affinity DataIC50:  4.70E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325897(2-(5-phenylpentyl)pyrido[2,3-d]pyrimidin-4(3H)-one...)
Affinity DataIC50:  5.90E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325919(2-(3-(4-methoxyphenoxy)propoxy)pyrido[2,3-d]pyrimi...)
Affinity DataIC50:  6.30E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325901(2-(6-phenylhexyl)pyrido[2,3-d]pyrimidin-4(3H)-one ...)
Affinity DataIC50:  1.90E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325913(2-(3-(2-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataIC50:  3.30E+4nMAssay Description:Displacement of radioligand from human GPR109BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325903(2-(7-phenylheptyl)pyrido[2,3-d]pyrimidin-4(3H)-one...)
Affinity DataIC50:  4.80E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325906(2-(3-phenoxypropyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325905(2-benzylpyrido[2,3-d]pyrimidin-4(3H)-one | CHEMBL1...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325922(2-((4-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325898(2-phenethylpyrido[2,3-d]pyrimidin-4(3H)-one | CHEM...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325902(2-(3-phenylpropyl)pyrido[2,3-d]pyrimidin-4(3H)-one...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of radioligand from human GPR109BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325924(2-((3-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at rat GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325922(2-((4-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at rat GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325924(2-((3-chlorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataEC50:  340nMAssay Description:Agonist activity at human GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325922(2-((4-fluorophenethyloxy)methyl)pyrido[2,3-d]pyrim...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325913(2-(3-(2-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325913(2-(3-(2-chlorophenoxy)propoxy)pyrido[2,3-d]pyrimid...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at rat GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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