Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50032388
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328434(3-bromo-N-(4-morpholinophenyl)-6-(pyridin-3-yl)imi...)
Affinity DataIC50:  152nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328436(3-chloro-N-(4-morpholin-4-ylphenyl)-6-pyridin-3-yl...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328433(3-methyl-N-(4-morpholinophenyl)-6-(pyridin-3-yl)im...)
Affinity DataIC50:  208nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase C(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328436(3-chloro-N-(4-morpholin-4-ylphenyl)-6-pyridin-3-yl...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of human aurora CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328421(CHEMBL1257211 | N-(4-morpholinophenyl)-6-(pyridin-...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328424(CHEMBL1257333 | N-(4-(6-(pyridin-3-yl)imidazo[1,2-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328422(CHEMBL1257331 | N-(4-methoxyphenyl)-6-(pyridin-3-y...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328425(CHEMBL1257445 | N-(4-(6-(pyridin-3-yl)imidazo[1,2-...)
Affinity DataIC50:  3.75E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328435(CHEMBL1258604 | N-(4-morpholinophenyl)-3,6-di(pyri...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328432(CHEMBL1258379 | N-(3-(8-(4-methoxyphenylamino)imid...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328427(6-(3-aminophenyl)-N-(4-methoxyphenyl)imidazo[1,2-a...)
Affinity DataIC50:  5.48E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328423(CHEMBL1257332 | N-(4-chlorophenyl)-6-(pyridin-3-yl...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328431(4-methoxy-N-(3-(8-(4-methoxyphenylamino)imidazo[1,...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328420(CHEMBL1257210 | N-phenyl-6-(pyridin-3-yl)imidazo[1...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328429(1-(3-(8-(4-methoxyphenylamino)imidazo[1,2-a]pyrazi...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328428(2-methoxy-N-(3-(8-(4-methoxyphenylamino)imidazo[1,...)
Affinity DataIC50:  7.31E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328430(1-(4-methoxyphenyl)-3-(3-(8-(4-methoxyphenylamino)...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328426(CHEMBL1257923 | N-(4-methoxyphenyl)-6-(1-methyl-1H...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of human aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50328437(CHEMBL1230687 | N-(3-(3-chloro-8-(4-morpholinophen...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed