Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50032423
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.18nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(N,N'-(Iminodinonane-9,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataEC50:  1.34nMAssay Description:Antagonist activity at rat brain CB1 receptor assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(N,N'-[(Methylimino)dipentane-5,1-diyl]bis[5-(4-chl...)
Affinity DataEC50:  1.78nMAssay Description:Antagonist activity at rat brain CB1 receptor assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(N-{11-[(11-Aminoundecyl)amino]undecyl}-5-(4-chloro...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(N,N'-(Iminodiheptane-7,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  4.41nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(N-{11-[(11-Aminoundecyl)amino]undecyl}-5-(4-chloro...)
Affinity DataKi:  4.56nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(N-{9-[(9-Aminononyl)amino]nonyl}-5-(4-chlorophenyl...)
Affinity DataKi:  5.44nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328967(N-{11-[(11-Aminoundecyl)(methyl)amino]undecyl}-5-(...)
Affinity DataKi:  5.51nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(N-{9-[(9-Aminononyl)(methyl)amino]nonyl}-5-(4-chlo...)
Affinity DataKi:  6.12nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  6.18nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(N,N'-[(Methylimino)dipentane-5,1-diyl]bis[5-(4-chl...)
Affinity DataKi:  6.35nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(N-{9-[(9-Aminononyl)(methyl)amino]nonyl}-5-(4-chlo...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(N,N'-(Iminodiheptane-7,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(N-{9-[(9-Aminononyl)amino]nonyl}-5-(4-chlorophenyl...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328967(N-{11-[(11-Aminoundecyl)(methyl)amino]undecyl}-5-(...)
Affinity DataKi:  14.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328961(N-{7-[(7-Aminoheptyl)(methyl)amino]heptyl}-5-(4-ch...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328965(N,N'-[(Methylimino)diheptane-7,1-diyl]bis[5-(4-chl...)
Affinity DataKi:  17.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328958(N-{7-[(7-Aminoheptyl)amino]heptyl}-5-(4-chlorophen...)
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328965(N,N'-[(Methylimino)diheptane-7,1-diyl]bis[5-(4-chl...)
Affinity DataKi:  27.5nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(N,N'-(Iminodinonane-9,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataEC50:  27.9nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328963(N,N'-[(Methylimino)diundecane-11,1-diyl]bis[5-(4-c...)
Affinity DataEC50:  29.3nMAssay Description:Antagonist activity at rat brain CB1 receptor assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(N,N'-(Iminodipentane-5,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  30.4nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(N,N'-(Iminodipentane-5,1-diyl)bis[5-(4-chloropheny...)
Affinity DataEC50:  33nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328950(N,N'-(Iminodiundecane-11,1-diyl)bis[5-(4-chlorophe...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328961(N-{7-[(7-Aminoheptyl)(methyl)amino]heptyl}-5-(4-ch...)
Affinity DataKi:  37.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(N,N'-[(Methylimino)dipentane-5,1-diyl]bis[5-(4-chl...)
Affinity DataKi:  38.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(N,N'-(Iminodipropane-3,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  41.9nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328958(N-{7-[(7-Aminoheptyl)amino]heptyl}-5-(4-chlorophen...)
Affinity DataKi:  46.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(N,N'-(Iminodinonane-9,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataKi:  54.1nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328951(N,N'-(Iminodinonane-9,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataKi:  57.4nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328966(N,N'-[(Methylimino)dipentane-5,1-diyl]bis[5-(4-chl...)
Affinity DataEC50:  59.8nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328953(N,N'-(Iminodipentane-5,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  68.1nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(N,N'-(Iminodipropane-3,1-diyl)bis[5-(4-chloropheny...)
Affinity DataEC50:  84.2nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328962(N-{5-[(5-Aminopentyl)(methyl)amino]pentyl}-5-(4-ch...)
Affinity DataKi:  88.8nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(N,N'-(Iminodiethane-2,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328964(N,N'-[(Methylimino)dinonane-9,1-diyl]bis[5-(4-chlo...)
Affinity DataKi:  94.1nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328950(N,N'-(Iminodiundecane-11,1-diyl)bis[5-(4-chlorophe...)
Affinity DataKi:  99.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328964(N,N'-[(Methylimino)dinonane-9,1-diyl]bis[5-(4-chlo...)
Affinity DataEC50:  161nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328962(N-{5-[(5-Aminopentyl)(methyl)amino]pentyl}-5-(4-ch...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328954(N,N'-(Iminodipropane-3,1-diyl)bis[5-(4-chloropheny...)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328952(N,N'-(Iminodiheptane-7,1-diyl)bis[5-(4-chloropheny...)
Affinity DataEC50:  179nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(N,N'-(Iminodiethane-2,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328959(N-{5-[(5-Aminopentyl)amino]pentyl}-5-(4-chlorophen...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328955(N,N'-(Iminodiethane-2,1-diyl)bis[5-(4-chlorophenyl...)
Affinity DataEC50:  237nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328964(N,N'-[(Methylimino)dinonane-9,1-diyl]bis[5-(4-chlo...)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328960(N-{9-[(9-Aminononyl)(methyl)amino]nonyl}-5-(4-chlo...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328956(N-{11-[(11-Aminoundecyl)amino]undecyl}-5-(4-chloro...)
Affinity DataKi:  305nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328959(N-{5-[(5-Aminopentyl)amino]pentyl}-5-(4-chlorophen...)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50328957(N-{9-[(9-Aminononyl)amino]nonyl}-5-(4-chlorophenyl...)
Affinity DataKi:  419nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
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