Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50034290
TargetCannabinoid receptor 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360023(CHEMBL1928337)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360023(CHEMBL1928337)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataKi:  7.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360022(CHEMBL1928336)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360021(CHEMBL1164701)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50360021(CHEMBL1164701)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM85515(Ampyrone | CAS_83-07-8 | EN300-17058 | NSC_2151 | ...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM85515(Ampyrone | CAS_83-07-8 | EN300-17058 | NSC_2151 | ...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T

Curated by ChEMBL
LigandPNGBDBM50054471((5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed